Search results for "2307 Health"

showing 3 items of 3 documents

Spectrum of styrene-induced DNA adducts: the relationship to other biomarkers and prospects in human biomonitoring.

2002

Styrene is an important industrial chemical that has shown genotoxicity in many toxicology assays. This is believed to be related to the DNA-binding properties of styrene-7,8-oxide (SO), a major metabolite of styrene. In this review, we have summarized knowledge on various aspects of styrene genotoxicity, especially in order to understand the formation and removal of primary DNA lesions, and the usefulness of biomarkers for risk assessment. Biological significances of specific DNA adducts and their role in the cascade of genotoxic events are discussed. Links between markers of external and internal exposure are evaluated, as well as metabolic aspects leading to the formation of DNA adducts …

Health Toxicology and MutagenesisMetabolitePopulation10050 Institute of Pharmacology and Toxicology610 Medicine & healthBiologyIn Vitro Techniquesmedicine.disease_causeRisk AssessmentStyrenechemistry.chemical_compoundDNA Adducts1311 GeneticsOccupational ExposureBiomonitoring2307 Health Toxicology and MutagenesisGeneticsmedicineAnimalsHumanseducationStyreneGeneticseducation.field_of_studyPrimary (chemistry)Binding SitesDNAchemistryBiochemistry570 Life sciences; biologyEpoxy CompoundsXenobioticGenotoxicityDNABiomarkersEnvironmental MonitoringMutagensMutation research
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Xenobiotic-metabolizing enzyme activities in hybrid cell lines established by fusion of primary rat liver parenchymal cells with hepatoma cells

1992

1. The activities of xenobiotic-metabolizing enzymes were determined in hybrid cell lines (hepatocytoma, HPCT) which have been established by fusion of liver parenchymal cells from adult rat (PC) with cells from a Reuber hepatoma cell line (FAO). 2. Cytochrome P450 was not measurable spectrophotometrically in FAO and HPCT. P450-dependent conversion of testosterone was below the detection limit in FAO and only marginally present in HPCT. 3. Microsomal and cytosolic epoxide hydrolase, glutathione S-transferase and phenol sulphotranserase were low or even below detection limit in FAO. These enzyme activities were significantly higher in HPCT and correspond to about 1-10% the activities measure…

Male1303 BiochemistryHealth Toxicology and Mutagenesis10050 Institute of Pharmacology and Toxicology610 Medicine & healthHybrid CellsToxicologyBiochemistryCell LineMixed Function OxygenasesXenobioticsCell FusionRats Sprague-Dawleychemistry.chemical_compoundLiver Neoplasms Experimental2307 Health Toxicology and MutagenesisTumor Cells CulturedAnimalsEnzyme inducerEpoxide hydrolasePharmacologychemistry.chemical_classificationbiologydigestive oral and skin physiologyCytochrome P4503005 ToxicologyGeneral MedicineGlutathioneRatsEnzyme3004 PharmacologychemistryBiochemistryLiverCell cultureEnzyme inhibitorbiology.proteinMicrosome570 Life sciences; biology
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cis- and trans-1,2-diphenylaziridines: induction of xenobiotic-metabolizing enzymes in rat liver and mutagenicity in Salmonella typhimurium.

1986

trans-Stilbene imine (trans-1,2-diphenylaziridine) is the nitrogen analog of trans-stilbene oxide, a potent inducer of several microsomal and cytosolic xenobiotic-metabolizing enzymes. Although the acute toxicity of cis- and trans-stilbene imines prevents their application at the usual dose for trans-stilbene oxide (400 mg/kg/day), it is apparent that the imines nevertheless potently induce several xenobiotic-metabolizing enzymes in rat liver. The IP administration of trans-stilbene imine resulted in statistically significant increases in the activities of aminopyrine N-demethylase, microsomal epoxide hydrolase, glutathione transferase (toward 1-chloro-2,4-dinitrobenzene, 1,2-dichloro-4-nit…

MaleSalmonella typhimuriumStereochemistryHealth Toxicology and MutagenesisImineAziridines10050 Institute of Pharmacology and Toxicology610 Medicine & healthMutagenToxicologymedicine.disease_causeAmes testchemistry.chemical_compound2307 Health Toxicology and MutagenesismedicineAnimalsToxicology and MutagenesisEnzyme inducerchemistry.chemical_classificationbiologyAzirinesMutagenicity Tests3005 ToxicologyRats Inbred StrainsStereoisomerismGeneral MedicineCis trans isomerizationRatsEnzymechemistryBiochemistryLiverHealthMicrosomal epoxide hydrolaseEnzyme InductionMicrosomebiology.protein570 Life sciences; biologyMutagensArchives of toxicology
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